Virtual Screening and ADMET Studies to Identify KSP Inhibitors as Anticancer Therapeutics
نویسندگان
چکیده
منابع مشابه
Virtual Screening and ADMET studies to identify KSP inhibitors as anticancer therapeutics
Introduction Kinesin spindle protein (KSP), also known as Hs Eg5 has emerged as a promising target for a new generation antimitotic chemotherapeutic agents, it is a member of the kinesin superfamily of molecular motors that utilize the energy generated from the hydrolysis of ATP to transport vesicles, organelles, and microtubules [1-3]. Ispinesib has emerged as a potent KSP inhibitor with sub n...
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ژورنال
عنوان ژورنال: International Journal of Advances in Pharmaceutical Sciences
سال: 2017
ISSN: 0976-1055
DOI: 10.5138/09761055.2069